Key Takeaways

  • Check apical pulse for 1 minute before digoxin; hold if HR < 60 in adults
  • Warfarin is monitored by PT/INR; heparin is monitored by aPTT
  • Rinse mouth after using inhaled corticosteroids to prevent thrush
  • Assess respiratory rate before opioids; hold if RR < 12
  • Insulin: clear before cloudy when mixing; never mix long-acting insulins
Last updated: January 2026

Common Drug Classifications

Understanding drug classifications, their mechanisms, and nursing implications is essential for safe medication administration. This section covers major drug classes commonly encountered in LPN/VN practice.

Cardiovascular Medications

Antihypertensives

ClassExamplesMechanismKey Nursing Points
ACE Inhibitors (-pril)Lisinopril, enalaprilBlock angiotensin II formationMonitor for dry cough, hyperkalemia, first-dose hypotension
ARBs (-sartan)Losartan, valsartanBlock angiotensin receptorsSimilar to ACE inhibitors but less cough
Beta Blockers (-olol)Metoprolol, atenololDecrease HR and contractilityMonitor HR (hold if <60), assess for fatigue, mask hypoglycemia
Calcium Channel Blockers (-dipine)Amlodipine, diltiazemVasodilation, decrease contractilityMonitor BP, assess for edema, constipation
DiureticsHCTZ, furosemideIncrease urine outputMonitor electrolytes (K+), I&O, weight

Cardiac Glycosides

Digoxin:

  • Increases cardiac contractility (positive inotrope)
  • Decreases heart rate (negative chronotrope)
  • Therapeutic range: 0.5-2.0 ng/mL
  • Hold if: HR < 60 (adult), < 90-100 (infant)
  • Toxicity signs: Anorexia, nausea, visual disturbances (halos), bradycardia, arrhythmias
  • Monitor potassium (hypokalemia increases toxicity risk)

Anticoagulants

DrugMonitoringAntidote
HeparinaPTT (1.5-2.5× normal)Protamine sulfate
Enoxaparin (Lovenox)Anti-Xa levels (if monitored)Protamine sulfate (partial)
Warfarin (Coumadin)PT/INR (2.0-3.0 for most)Vitamin K, fresh frozen plasma

Respiratory Medications

ClassExamplesPurposeNursing Points
Short-acting bronchodilators (SABA)AlbuterolAcute bronchospasm reliefRapid onset (rescue inhaler), may cause tachycardia
Long-acting bronchodilators (LABA)SalmeterolMaintenance therapyNot for acute attacks, use with ICS for asthma
Inhaled corticosteroids (ICS)Fluticasone, budesonideReduce inflammationRinse mouth after use, prevents thrush
AnticholinergicsIpratropium, tiotropiumBronchodilationDry mouth common, avoid in glaucoma

Gastrointestinal Medications

ClassExamplesPurposeNursing Points
Proton Pump Inhibitors (PPIs)Omeprazole, pantoprazoleReduce acid secretionTake 30-60 min before meals, long-term use risks
H2 BlockersFamotidine, ranitidine*Reduce acidLess potent than PPIs
AntacidsCalcium carbonate, aluminum hydroxideNeutralize acidTake 1-3 hours after meals, drug interactions
AntiemeticsOndansetron, promethazinePrevent/treat nauseaMay cause drowsiness, ondansetron: check QT
LaxativesSenna, docusate, bisacodylPromote bowel movementsAdequate fluids, don't use long-term

*Note: Ranitidine recalled; famotidine is alternative

Endocrine Medications

Insulins

TypeOnsetPeakDurationExample
Rapid-acting10-30 min30 min-3 hr3-5 hrLispro (Humalog), Aspart (NovoLog)
Short-acting30-60 min2-4 hr5-8 hrRegular (Humulin R)
Intermediate1-2 hr4-12 hr12-18 hrNPH (Humulin N)
Long-acting1-2 hrMinimal/none24+ hrGlargine (Lantus), Detemir (Levemir)

Insulin Administration:

  • Always verify dose with another nurse
  • Rotate injection sites within same region
  • Clear insulins before cloudy when mixing
  • Do NOT mix long-acting with other insulins
  • Store open vials at room temp (28 days); unopened in refrigerator

Oral Antidiabetic Agents

ClassExampleMechanismKey Points
BiguanidesMetforminDecreases glucose productionHold before contrast dye, no alcohol
SulfonylureasGlipizide, glyburideStimulate insulin releaseRisk of hypoglycemia, take with meals
DPP-4 InhibitorsSitagliptinIncrease incretin levelsLow hypoglycemia risk

Pain Medications

Opioid Analgesics

DrugEquianalgesic DoseKey Points
Morphine10 mg IV/30 mg POStandard for comparison
Hydromorphone (Dilaudid)1.5 mg IV/7.5 mg PO4-5× more potent than morphine
Fentanyl100 mcg IVVery potent, rapid onset
Oxycodone20 mg POOral only, often combined with APAP

Nursing Considerations:

  • Assess respiratory rate before administration (hold if RR <12)
  • Monitor sedation level
  • Constipation is expected; implement bowel regimen
  • Assess pain before and after administration
  • Know location of naloxone (Narcan) for reversal

Non-Opioid Analgesics

DrugMaximum Daily DoseKey Points
Acetaminophen3-4 g/day (less with liver disease)Hepatotoxic in overdose
Ibuprofen (NSAID)3.2 g/dayGI bleeding risk, renal effects
Ketorolac (NSAID)5 days maxVery effective, significant GI/renal risks

Neurological Medications

ClassExamplesPurposeNursing Points
BenzodiazepinesLorazepam, diazepamAnxiety, seizures, sedationRespiratory depression, fall risk, flumazenil reverses
AntiepilepticsPhenytoin, valproic acid, levetiracetamSeizure preventionMonitor levels (phenytoin: 10-20 mcg/mL), CBC
SSRIsSertraline, fluoxetineDepression, anxiety2-4 weeks for effect, serotonin syndrome risk
Test Your Knowledge

Before administering digoxin, what assessment should the LPN/VN perform?

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D
Test Your Knowledge

A patient is taking warfarin. Which laboratory value should the LPN/VN monitor?

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B
C
D
Test Your Knowledge

Which insulin has the longest duration of action?

A
B
C
D